| Intro |
8:30 |
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Welcome speech, practical information |
Session 1
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Chairman: Prof. Martin Doležal Co-chairman: Prof. Jarmila Vinšová |
| PL-1 |
8:40 |
Petr Zimčík |
Advances in the use of phthalocyanines and their analogues in photodynamic therapy |
| SC-1 |
9:00 |
Veronika Vyletelová |
Modifications of HDL components´ gene expression in liver of rat with adjuvant arthritis |
| SC-2 |
9:15 |
Mária Nováková |
Effect of heat-killed lactobacilli on the expression of genes related to lipid metabolism and inflammation |
| SC-3 |
9:30 |
Martina Mušković |
Synthesis, photophysical, photochemical and photobiological properties of amphiphilic Zn(II) and free base tripyridylporphyrins |
| SC-4 |
9:45 |
Eva Havránková |
Triazinyl-substituted benzenesulfonamides as inhibitors of bacterial carbonic anhydrase |
| break |
10:00 |
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Session 2
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Chairman: Prof. Jarmila Vinšová Co-chairman: Prof. Petr Zimčík |
| PL-2 |
10:15 |
Markus Pietsch |
Targeting tumor-relevant proteins – Inhibitors of the subunit interaction of protein kinase CK2 |
| SC-5 |
10:45 |
Martin Vrbický |
Synthesis of oxazolidinone drugs Linezolid and Rivaroxaban via asymmetric Henry reaction |
| SC-6 |
11:00 |
Vinod S.K. Pallabothula |
Design, synthesis, SAR and in silico studies of 3-aminopyrazine-2-carboxamides as antimicrobials |
| SC-7 |
11:15 |
Marek Kerda |
Synthesis of hydrophilic substituted 3-benzamidopyrazine-2-carboxamides and docking into a homology model of mycobacterial prolyl-tRNA synthetase |
| SC-8 |
11:30 |
Aljoša Bolje |
Structural characterization and stability of proteins in solid forms |
| break |
11:45 |
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Session 3
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Chairman: Prof. Petr Zimčík Co-chairman: Assoc. Prof. Miroslav Miletín |
| PL-3 |
12:15 |
Reik Loeser |
Development of radiotracers as activity-based probes for the detection and imaging of transglutaminase 2 |
| SC-9 |
13:00 |
Jana Čurillová |
Physico-chemical and biological characterisation of novel derivatives containing N-arylpiperazine fragment |
| SC-10 |
13:15 |
Petr Šlechta |
Design, synthesis and preliminary biological evaluation of new boronic acids derivatives |
| SC-11 |
13:30 |
Bianka Oboňová |
Synthesis and analysis of bidentate Schiff bases as potential ligands for new metal complexes |
| break |
13:45 |
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Session 4
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Chairman: Assoc. Prof. Miroslav Miletín Co-chairman: Dr. Marta Kučerová |
| PL-4 |
14:00 |
Bohumír Grűner |
Boron clusters as newly emerging 3D platform for design of specific inhibitors of pharmaceutically relevant enzymes |
| SC-12 |
14:45 |
Magdaléna Onuščáková |
Synthesis and antiproliferative activity of selected N-hydroxycinnamamide derivates |
| SC-13 |
15:00 |
Veronika Ballayová |
Synthesis of Schiff bases with potential therapeutic activity |
| SC-14 |
15:15 |
Daria Nawrot |
Hybrid compounds containing 4-aminosalicylic acid as potential antituberculotics |
| break |
15:30 |
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Session 5
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Chairman: Dr. Marta Kučerová Co-chairman: Assoc. Prof. Jan Zitko |
| PL-5 |
15:45 |
Mark Olsen |
ASPH inhibitors for the treatment of metastatic cancer |
| SC-15 |
16:30 |
Peter Zubáč |
Design, synthesis and structure-based optimization of potential phenothiazine antimicrobials |
| SC-16 |
16:45 |
Negar Maafi |
Antimicrobial activity of semisynthetic derivatives of montanine-type alklaoids |
| SC-17 |
17:00 |
Rudolf Vrabec |
Indole alkaloid from Vinca minor L. with promising activity against Alzheimer's disease |
| break |
17:15 |
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Session 6
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Chairman: Dr. Marta Kučerová Co-chairman: Assoc. Prof. Jan Zitko |
| PL-6 |
17:30 |
Roman Dembinski |
Synthesis of modified nucleosides, derived from pyrimidine, and their biological properties |
| End |
18:00 |
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